
H-9 hydrochloride
CAS No. 116970-50-4
H-9 hydrochloride( —— )
Catalog No. M21838 CAS No. 116970-50-4
H-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM).
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
10MG | 76 | In Stock |
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50MG | 320 | In Stock |
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100MG | Get Quote | In Stock |
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200MG | Get Quote | In Stock |
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500MG | Get Quote | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameH-9 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionH-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM).
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DescriptionH-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM). It has shown to dramatically reduce the GABA response of GABAA currents in retinal rod bipolar cells as well as inhibit smooth muscle cell relaxation induced by cGRP. H-9 dihydrochloride has also been used for purification of protein kinases in ligand affinity chromatography.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorcGKI
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Research Area——
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Indication——
Chemical Information
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CAS Number116970-50-4
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Formula Weight287.77
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Molecular FormulaC11H13N3O2S?HCl
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Purity>98% (HPLC)
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Solubility——
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SMILESC1=CC2=C(C=CN=C2)C(=C1)S(=O)(=O)NCCN.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wolf, M., et al. 1985. J. Biol. Chem. 260: 15718-15722. PMID: 4066694
2. Inagaki, M., et al. 1985. J. Biol. Chem. 260: 2922-2925. PMID: 2982842
3. Gillette, M.A., et al. 1996. J. Neurophysiol. 76: 3070-3086. PMID: 8930256
molnova catalog



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